Onye ntanye (ratelgravir) bụ onye na- eme ihe na-eme ihe na-eme ihe na-eme ka ọgwụ nje nje na-agwọ ọrịa HIV . Nwaanyị ahụ bụ onye mmegide nke mbụ iji nweta nkwado site n'aka US Food and Drug Administration (FDA).
N'October 2007, e nyere ikikere maka iji ndị okenye na- eguzogide ọgwụ mgbochi ndị ọzọ . Ma site na July 2009, na mgbe e mesịrị na Disemba 2011, FDA gbasaa ihe ngosi ya, na-enye ohere maka ndị okenye niile na-ebute nje HIV, yana ụmụaka dị afọ 2-18.
Nwaanyị nọ n'etiti ọgwụ ndị a na-atụ aro ugbu a dịka nhọrọ kachasị maka ọnụọgụ nje HIV na US
Usoro
Nwanyị nwanyị dị na ụdị anọ dị iche iche:
- Maka ụmụaka okenye na ụmụaka toro eto, enwere nwa mpempe akwụkwọ dị ka mpempe akwụkwọ mpịakọta 400mg, oval na ọdịdị na pink-oma na agba. Ọnụ ọgụgụ "207" dị na otu akụkụ.
- Maka ụmụaka na-enweghị ike iji mbadamba nkume, Iche akwụkwọ dị dị ka 100mg chewable (oval, beige, nke nwere "477," nke gbanwere maka nkewa) ma ọ bụ 25mg chewable (acha odo odo, gburugburu, nke nwere "473" "). Ha abụọ bụ orange-banana flavored.
- Maka obere ụmụaka na-enweghị ike ịme ihe dị mma, Ntinye akwụkwọ dị na otu mkpọ, 100mg nkwupụta ụlọnga. Akwụsịtụ ụlọnga na-ejikọta ya na 5mL mmiri ma na-ejikwa serring serial. Ozugbo agwakọta ya, a ga-eji nkwadebe okwu ọnụ mee ihe n'ime nkeji iri atọ, ya na ihe ọ bụla furu efu ozugbo tụfuuru ya. Akwụsịtụsịsịsịsịsịsị na-echere banana.
Ejila dochie anya onye isi ụlọ ma ọ bụ nkwupụta ụlọnga maka nkwupụta ụda nke ihe nkiri na-ekpuchi Filiks dịka nchịkọta ndị ahụ abụghị usoro ndụ. Jiri naanị dị ka a gwara gị (lee anya n'okpuru ebe a).
Ngwunye
Akwụsị 400mg, ihe mbadamba ihe nkiri a ga-edere maka ndị okenye na maka ụmụaka toro eto nwere ike ilo mbadamba, dị ka ndị a:
- Ndị okenye: otu mbadamba 400mg, were ugboro abụọ kwa ụbọchị
- Maka ụmụaka ma ọ bụ na-eto eto 55 pound (25kg) ma ọ bụ n'elu: otu 400mg mbadamba, were ugboro abụọ kwa ụbọchị
A ga-edebere mbadamba nkume dị iche iche nke na -edozi ahụ maka ụmụaka na-eru kilogram iri abụọ (20kg) ma ọ bụ karịa ndị na-enweghị ike ilo mbadamba, dị ka ndị a:
- 44 pound (20kg) na-erughị pasent 62 (28kg): 150mg ugboro abụọ kwa ụbọchị
- 62 kilogram (28kg) na-erughị 88 pound (40kg): 200mg ugboro abụọ kwa ụbọchị
- Ihe karịrị 88 kilogram (40kg): 300mg ugboro abụọ kwa ụbọchị
A ghaghị idebe nkwonkwo ụbụrụ na-edozi ahụ ma ọ bụ mbadamba ụrọ maka ụmụaka na-atụ egwu ma ọ dịkarịa ala kilogram (3kg) na-erughị 55 kilogram (25kg), dị ka ndị a:
- 6.5 pound (3kg) na-erughị 8,8 paụnd (4kg): 1mL (20mg) kwadebere nkwonkwo ụlọnga ugboro abụọ kwa ụbọchị
- Akara 8kg) na-erughị kilogram iri isii (6kg): 1.5mL (30mg) kwadebere nkwupụta ụlọnga ebubo ugboro abụọ kwa ụbọchị
- Pound (6kg) na-erughị kilogram 17 (8kg): 2mL (40mg) kwadebere nkwupụta ụlọnga nke okpukpu abụọ ugboro abụọ
- 17 kilogram (8kg) na ihe na-erughị kilogram 24 (11kg): 3mL (60mg) kwadebere nkwụmkpụ ụra ugboro abụọ kwa ụbọchị
- 24 kilogram (11kg) na ihe na-erughị kilogram 30 (14kg): 4mL (80kg) kwadebere nkwụmkpụ ụra ugboro abụọ kwa ụbọchị 75 ma ọ bụ 75 mg e nwere ike iji chetable.
- 30 kilogram (14kg) na ihe na-erughị kilogram iri abụọ (20kg): 5mL (100kg) kwadebere nkwupụta ụlọnga ebubo ugboro abụọ kwa ụbọchị ma ọ bụ 100mg mbadamba ụrọ e ugboro abụọ kwa ụbọchị
Nchịkọta Ọgwụ
Enwere ike iji nri ma ọ bụ na-enweghị nri. Enwereghi ike iburu onye na-esote nwa ya n'onwe ya ma kwesiri idebe ya dika akụkụ nke ọgwụgwọ antiretroviral (cART) .
Mmetụta Na-agakarị
Ihe kachasị emetụtakwa (nke mere na 2% ma ọ bụ obere nke ikpe) bụ:
- Mkpụrụ obi
- Isi ọwụwa
- Dizziness
- Nausea
- Ike ọgwụgwụ
Contraindications
Ọ dịghị
Mmekọrịta Ọgwụ Drug-Drug
Biko nye dọkịta gị ndụmọdụ ma ọ bụrụ na ị na-ewere ọgwụ ọ bụla dịka a naghị atụ aro ka ha na-elekọta gị na Nwaanyị ahụ nwere ike igbochi ịme ọgwụ:
- Ngwọrọgwu Rifampin dabeere na Rifampin: Rifadan, Rifater, Rifamate, Rimactane
- Aluminum- ma ọ bụ magnetium dabeere na antacids (dịka, Tums, Mmiri nke Magnesia, wdg.)
Echiche
Ndị ọrịa nwere ahụmahụ na- adighi ahụ mgbe ịmalite Isentress kwesịrị ịkpọtụrụ dọkịta ha ozugbo. A ghaghị ịkwụsị ọgwụgwọ ma gwọọ ọgwụgwọ ma ọ bụrụ na ọkụ ọkụ na-esonyere ya na ahụ ọkụ, nkwonkwo ma ọ bụ nkwonkwo ahụ, ọnyá ma ọ bụ ọnyá, ọbara ọbara ma ọ bụ ọzịza nke anya, ikpu nke ihu ma ọ bụ ọnụ, ma ọ bụ nsogbu iku ume. Ọrịa ndị na-ahụtụbeghị mmeghachi omume nke ịmalite ịmalite ịmalite ịmịnye nwa nwanyị ekwesịghị ịbụ onye a na-agbagha ya na ọgwụ ahụ mgbe ọ kwụsịrị ihe mgbaàmà.
Nnyocha ụmụ anụmanụ egosighi na ọ bụ nwa ebu n'afọ ma ọ bụ nwa ebu n'afọ n'oge ime nwa na ụmụ oke ma ọ bụ rabbits ekpughere nye nwanyị. Otú ọ dị, enwebeghị ike imetụta mmetụta nke nwa nwanyị na-enye nwa ara, na, n'ihi ya, a dịghị enye aro maka ndị nne na-ebute Nwaanyị.
Isi mmalite:
Ngalaba Ahụike na Ọrụ Ndị Mmadụ (DHHS). "Ntuziaka Maka Eji Ndị Na-akpata Antiretroviral na HIV-1-Adults Adults and Adolescents." Rockville, Maryland.
FDA. "FDA na-amụbawanye Iji Ntube Ọrịa Na-ahụ Maka Ọrịa Na-ahụ Maka Ụmụaka na Ọkaakaa." Silver Spring, Maryland; December 21, 2011.
Reuters. "Kwadoo OKWU 2-FDA tinyekwuo nke Merkel's Isentress HIV Drug." July 9, 2009.
Nchịkwa nri na ọgwụgwọ US (FDA). "Ngwakọta ngwongwo ngwongwo - Ngwá ọgwụ: Anentressress (ratelgravir) 400mg Mbadamba." Silver Spring, Maryland; October 12, 2007.